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Journal Articles Tetrahedron Year : 2014

A convergent route to functional protected amines, diamines, and β-amino acids

Abstract

Phthalimide protected amines react with NBS under peroxide initiation to give geminal phthalimido-bromo derivatives, which are readily converted into the corresponding xanthates. These xanthates in turn undergo radical additions to numerous olefins, providing a convergent and modular access to densely functionalized protected amines and diamines.
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hal-01082412 , version 1 (13-11-2014)

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Songzhe Han, Rachel A. Jones, Béatrice Quiclet-Sire, Samir Z. Zard. A convergent route to functional protected amines, diamines, and β-amino acids. Tetrahedron, 2014, 70 (40), pp.7192-7206. ⟨10.1016/j.tet.2014.07.055⟩. ⟨hal-01082412⟩
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